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Isoform-Selective ATAD2 Chemical Probe with Novel Chemical Structure and Unusual Mode of Action

October 18, 2017

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Structural insight into allosteric modulation of protease-activated receptor 2

April 26, 2017

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Pharmacological property optimization for allosteric ligands: A medicinal chemistry perspective.

April 3, 2017

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Discovery of a potent BTK inhibitor with a novel binding mode using parallel selections with a DNA-encoded chemical library.

January 5, 2017

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Structure Based Design of Non-Natural Peptidic Macrocyclic Mcl-1 Inhibitors

December 27, 2016

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DNA-encoded chemistry: enabling the deeper sampling of chemical space.

December 9, 2016

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Discovery of cofactor-specific, bactericidal Mycobacterium tuberculosis InhA inhibitors using DNA-encoded library technology.

November 18, 2016

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Bromodomain inhibitors regulate the C9ORF72 locus in ALS

September 1, 2015

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Encoded Library Synthesis Using Chemical Ligation and the Discovery of sEH Inhibitors from a 334-Million Member Library.

June 10, 2015

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Chemical ligation methods for the tagging of DNA-encoded chemical libraries.

March 8, 2015